Histamine <sub>H4</sub>Receptor Research

COST Presentations in Meetings

Adami, M., Pozzoli, C., Smits, R., Leurs, R. and Coruzzi G. Gastric effects of histamine: any role for H4 receptors? XXXIV Meeting of the Italian Pharm Soc, Rimini, 14-17 October 2009
Alfón J, Ardanaz N, Gil B, Fernández A, Balsa D, Gómez L, Merlos M, Cortijo J, Morcillo E, Bartrolí X. UR-60427 a Novel H4 Receptor Inverse Agonist that Shows Good Efficacy in Rodent Asthma Models 38th European Histamine Research Society Meeting, Fulda (Germany), 13-16 May 2009
Alfón J., Gil B., Ardanaz N., Gómez-Valadés A. G., Mascaró C., González E., Motos A., Peña J., Porras M., Fernández A., Janer G., Giral M., Sánchez S., Gómez Ll.,
Balsa D., Cortijo J., Morcillo E., Bartroli J., Merlos M. UR-60427: First H4 receptor angagonist in preclinial development at Palau Pharma BioMedChem on Histamine H4 Receptor. New Compounds for Translational Steps, Frankfurt (Germany), 2009
Chazot P. H4R and sex steroids in salivary glands and Sjögren’s syndrome, British Soc for Pharmacology, 17.12.2009, London, UK
Chazot PL. COST Workshop Speaker “BioMed Chem on histamine H4 receptors: New compounds for translational step” Frankfurt, Germany October 2009
Chazot PL. Emerging Concepts in brain histamine – H3 and H4 histamine receptors in the CNS. Symposium Speaker SFN Conference Satellite Chicago, USA October 2009
Chazot PL. The CNS Histamine H3 and H4 receptors: molecular pharmacology, clinical applications and COST Action, July 2009, Speaker, Otago University School of Medical Sciences, NZ
Chazot PL. The Histamine H3 and H4 receptors: molecular pharmacology and clinical applications. July 2009, Speaker, Pfizer, Sandwich, UK
Clarke N, Brown C, Lane C, Mowbray C, Lim H, Leurs R, Schenck E, Perros-Huguet C, Yeadon M. Translation of species differences in histamine H4 pharmacology with PF-2988403 BPS winter meeting 2009, London, UK
Geschwandtner M*, Rossbach K, Bäumer W, Kietzmann M, Dijkstra D, Stark H, Werfel T, Gutzmer R. Murine and Human Langerhans Cells Express a Functional Histamine H4 Receptor: Modulation of Cell Migration and Function. 38th Annual Meeting of the European Histamine Research Society (EHRS), Fulda/Germany (May 13 -16, 2009), Abstract O29 (p. 53). ARTHUR A. HANCOCK YOUNG INVESTIGATOR AWARD 1ST PRIZE
Gutzmer R. The role of the histamine H4 receptor in chronic inflammatory skin disorders. BPS winter meeting 2009, London, UK
Handzlik J*, Kiec-Kononowicz K. Searching for histamine H4 receptor ligands among derivatives with N-methylpiperazine amide motif BPS Winter 09 symposium, 17th Dec 2009 London, UK
Karcz T*, Handzlik J, Lazewska D, Kottke T, Seifert R, Stark H, Kiec-Kononowicz K. Search for histamine H4 receptor ligands in the group of 4-methylpiperazino amide derivatives, 38th European Histamine Research Society Meeting, Fulda, Germany, 13-16 May, 2009
Kottke T*, Schneider E, Seifert R, Stark H. Functional Characterization of (1H-Imidazol-4-yl)alkyl Derivatives at Histamine H4 Receptor. 38th Annual Meeting of the European Histamine Research Society (EHRS), Fulda/Germany (May 13 -16, 2009), Abstract book P20 (p. 82).
Kuder KJ*, Kottke T, Stark H, Ligneau X, Camelin J-C, Seifert R, Kiec- Kononowicz K. Search for novel histamine H3/H4 receptors ligands in the group of (cyclic)isothiourea derivatives 2nd Polish Meeting on Medicinal Chemistry 8-10.09.09, Lublin, Poland
Kyriakidis K*, Zampeli E, Tiligada E. Effect of the H4 receptor antagonist JNJ7777120 on histamine levels of peripheral blood vessels in rats with adjuvant arthritis. Proceedings of the 38th Meeting of the European Histamine Research Society, 2009:52:?28 ARTHUR A. HANCOCK YOUNG INVESTIGATOR AWARD SPECIAL COMMENDATION
Leurs R. Recent advances in the molecular pharmacology of the H4 histamine receptor. BPS winter meeting 2009, London, UK
Moya-García A, Rodríguez C, Morillas I, Pino-Ángeles A, Fajardo I, García-Ranea JA, Sánchez-Jiménez F. Systemic approach to histamine receptor 4 activation. BPS winter meeting 2009, London, UK
Proschak E* et al. H4R Pseudoreceptor for homology model refinement and virtual screening. Meeting of WG4, Frankfurt, Germany, 2009, SL4.
Rayan A. The utility of intelligent learning engine for discovering novel H4 antagonists. International COST action workshop – BM0806 – WG4, 2009, Frankfurt, Germany
Rayan A. The utility of Intelligent Learning Engine in Drug Discovery Informatics. BPS winter meeting 2009, London, UK
Rivera ES. The H4 receptor and cancer pharmacology. BPS winter meeting 2009, London, UK
Roßbach K*, Stark H, Sander K, Kietzmann M, Bäumer W. Histamine H3 Receptor Antagonist-Induced Pruritus can be Inhibited by Blockade of Histamine H1 and H4 Receptors. 38th Annual Meeting of the European Histamine Research Society (EHRS), Fulda/Germany (May 2009), Abstract book P24 (p. 86).
Roßbach K*, Stark H, Sander K, Kietzmann M, Bäumer W. Histamine H3 Receptor Antagonist-Induced Pruritus can be Inhibited by Blockade of Histamine H1 and H4 Receptors. 11th Internatinal Congress of the European Association for Veterinary Pharmacology and Toxicology, Leipzig/Germany (July 12 – 16, 2009). J. Vet. Pharmacol. Ther. 2009, 32 (Suppl. 1), 220.
Sander K*, Kottke T, Proschak E, Tanrikulu Y, Schneider E, Seifert R, Schneider G, Stark H. Development of Diamininopyrimidines as Histamine H4 Receptor Ligands – Virtual Screening and Scaffold Optimisation. 38th Annual Meeting of the European Histamine Research Society (EHRS), Fulda/Germany (May 13 -16, 2009), Abstract O26 (p. 50). ARTHUR A. HANCOCK YOUNG INVESTIGATOR AWARD 2ND PRIZE
Sander K*, Kottke T, Tanrikulu Y, Proschak E, Schneider EH, Seifert R, Schneider G, Stark H. Functional Characterization of Diaminopyrimidines as Histamine H4 Receptor Ligands. Frontiers in Medicinal Chemistry, Barcelona/Spain (October 4-6, 2009). Drugs Fut. 2009, 34 (Suppl. A), 198 (PC.142).
Sasse A, Eleopra M, Stark H. Recent Advances in Histamine H4 Receptor Research, XVIIIth European Conference of GP2A "Groupement des Pharmacochimistes de l'Arc Atlantique" (GP2A), Trinity College Dublin, 3-4th, September 2009, Dublin, Ireland
Sasse A. Eleopra M, Stark H. Recent Advances in Histamine H4 Receptor Research. XVIIIth European Conference of GPA2 “Groupement des Pharmacochimistes de l'Arc Atlantique” (GP2A), Group of Medicinal Chemists of the Atlantic Arc, Trinity College Dublin/Ireland (September 3-4, 2009).
Stark H. Histamine Receptor Antagonists – From Bench to Bedside. 9th International Symposium on Pharmaceutical Sciences (ISOPS-9), Ankara/Turkey (June 23-26, 2009).
Stark H. Novel Histamine Receptor Ligands – From Bench to Bedside. Trinity College, Dublin/Ireland (September 18, 2009).
Stegaev V*, Chazot PL, Konttinen Y. H4R in murine and human salivary glands: effect of DHEA pro-hormone, Joint meeting of the Danish Stem Cell and Finnish Musculoskeleta PhD Graduate Schools, Odense, Denmark, 11.12.2009
Tiligada E Pharmacology and therapeutic perspective of the histamine H4 receptor: state-of-the-art, International COST Action BM0806 Workshop on BioMedChem on Histamine H4 Receptor-New Compounds for Translational Steps, Goethe-University, Biozentrum, Frankfurt am Main, Germany, 2009:11:PL1
Tiligada E. Pharmacology and therapeutic perspective of the histamine H4 receptor: state-of-the-art, “BioMedChem on Histamine H4 Receptor - New Compounds for Translational Steps”, COST Action BM0806 International WG4 Workshop, Johann Wolfgang Goethe-University, Frankfurt am Main, Germany, 6.10.2009
Wiecek M*, Kottke T, Ligneau X, Camelin J-C, Stark H, Seifert R, Schunack W, Kiec- Kononowicz K. 3-(1H-imidazol-4-yl)propyl carbamates as histamine H3/H4 receptor ligands, 2nd Polish Meeting on Medicinal Chemistry 8-10.09.09, Lublin, Poland
Zampeli E*, Kyriakidis K, Tiligada E. Differential effects of H1 and H4 receptor antagonists on the cartilage histamine content in rats with adjuvant arthritis. Proceedings of the 38th Meeting of the European Histamine Research Society, 2009:87:?25